GPCR Pharmacology Platform

New medicines are still found more than they are made. We're building the operating system that changes that — knowledge compounds, the unknown retreats, and the field moves from search to design. Come navigate the expanse with us.

The platform for GPCR pharmacology built on the data the field has been missing — and designed to turn its most consequential unknowns into decisions.

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Affinity tells you a molecule binds.

It doesn't tell you whether binding does anything.

The Problem

The industry's primary filter is affinity — a measure of how tightly a drug candidate binds to its target protein. It drives medicinal chemistry, computational design, and AI optimization alike.

A molecule can bind tightly and produce no biological effect. It can bind weakly and transform a patient's life. Affinity predicts neither.

The conformational engagement of a drug at its target — whether binding actually moves the receptor, and how — is the measurement that determines whether a candidate works. It is possible to measure. It has simply never been done systematically, at scale, and with the data infrastructure to make the results actionable.

The data doesn't exist. Kinovi exists to capture it — and make it decisive.

$7.7B

Spent by the top 20 pharmaceutical companies on clinical programs terminated in 2024 alone.

Deloitte, 2024

40–50%

Of all clinical trial failures are efficacy failures — the drug didn't work as the binding data suggested it would.

Drugs fail in the clinic for reasons that were never measured in the lab.

Until now.

The Platform

The platform runs three layers deep.
Start at the top.

Intelligence
FIELD
Free energy Inference of
Energetic Landscape Dynamics
The AI model that turns KORE into decisions. As the corpus grows, the model sharpens — predictions improve, unknowns retreat, and the field moves from search to design. The intelligence layer that makes every prior experiment more valuable than the last.
Data
KORE
Kinetics Of
Receptor Engagement
The accumulating kinetic and conformational corpus for GPCR pharmacology — the foundation of FIELD. Every measurement Kinovi generates enters KORE, authenticated and permanently traceable via Klyph™. The corpus that compounds.
Measurement
Conformational Dynamics Transduction
Confidynt
Graphene Field-Effect Transistor
Nanodisc Platform
A graphene-based bioelectronic sensing platform that detects conformational engagement directly — not as a proxy, not downstream. The only instrument capable of characterizing how a molecule moves a full-length, Velax™-reconstituted GPCR in real time.
Enables → Dyne™
Functional Signal Transduction
Fluxynt
Graphene Field-Effect Transistor
Nanovesicle Platform
A graphene field-effect transistor platform operating on full-length GPCRs reconstituted in Kosmion™ nanovesicles — measuring downstream signaling flux without cellular noise, endogenous receptor interference, or the ambiguity of cell-based assays.
Enables → Kos™
The instruments behind KORE.

Built to be used. Built to compound. Built to last.

Scientific Foundation

The science is peer-reviewed.

Selected from 50+ peer-reviewed publications.

Biosensors & Bioelectronics · 2025

Nondestructive Methodology with Discerning Fruit Freshness Biomarker Compounds Using Olfactory Receptor Nanodisc-Loaded Graphene Transistors

S.E. Seo, S. Cho, K.H. Kim, S. Lee, J. Lee, Y.K. Cha, Y.-S. Ryu, T.H. Park, H.S. Song, O.S. Kwon

Science Advances · 2024

A Pattern Recognition Artificial Olfactory System Based on Human Olfactory Receptors and Organic Synaptic Devices

H.W. Song, D. Moon, Y. Won, Y.K. Cha, J. Yoo, T.H. Park, J.H. Oh

ACS Sensors · 2024

Combinatorial Pattern Response of Bioelectronic Nose for the Detection of Real Nerve Agents

J. Yoo, D. Lee, S. Lee, S. Kang, H.I. Kim, Y.J. Jang, J. Kim, T.H. Park

Advanced Functional Materials · 2023

Bioelectronic Tongue for Identifying and Masking Bitterness Based on Bitter Taste Receptor Agonism and Antagonism

J.Y. Hwang, K.H. Kim, S.E. Seo, Y. Nam, S. Jwa, I. Yang, T.H. Park, O.S. Kwon, S.H. Lee

ACS Applied Materials & Interfaces · 2022

Ultrasensitive Bioelectronic Tongue Based on the Venus Flytrap Domain of a Human Sweet Taste Receptor

J. Jeong, Y.K. Cha, S.R. Ahn, J. Shin, Y. Choi, T.H. Park, S. Hong

ACS Nano · 2017

Dopamine Receptor D1 Agonism and Antagonism Using a Field-Effect Transistor Assay

S.J. Park, H. Yang, S.H. Lee, H.S. Song, C.S. Park, J. Bae, O.S. Kwon, T.H. Park, J. Jang

Intellectual Property
10+
Issued and pending patents across US and international jurisdictions — spanning nanomaterial sensing, field-effect transduction, biological detection, and biophysical electronics.
Services

Insight at three depths.
Start where your program needs you.

Tier 3
Kos
Functional transduction profiling
Cell-free downstream signaling from a GPCR reconstituted in Kosmion™ nanovesicles — without cellular noise, endogenous receptor interference, or the ambiguity of cell-based assays. The closest measurement to clinical reality short of the clinic itself.
Tier 2
Dyne
Conformational engagement profiling
Direct detection of the conformational signal a molecule drives at a full-length GPCR in a Velax™ nanodisc. Whether binding moves the receptor, how far, and with what kinetic character. The measurement that predicts whether a binder is an activator.
Tier 1
Takt
Kinetic binding profiling
kon, koff, KD, and residence time at any GPCR — primary target and antitarget panel in a single engagement, run on Velax™ validated nanodisc constructs, executed entirely within the United States. The first measurement that separates candidates with real binding kinetics from those that only look good on affinity alone.
In closed development
Quord
The next layer of the platform. Founding partners are shaping it now.
Request received — we'll be in touch.
About
Joseph Azzarelli, PhD
Co-founder & CEO, Kinovi®
MIT · Swager Lab · Chemical Sensing & Nanomaterials
Pfizer · Neuroscience Medicinal Chemistry
Numo Health · Co-founder
14 issued patents · 10 pending

Joseph began his career at Pfizer Neuroscience, working in medicinal chemistry on Alzheimer's and schizophrenia programs — synthesizing candidates, watching programs advance and fail, and developing a first-hand understanding of what the field measures and what it consistently misses. The question that stayed with him: what was never measured?

He went on to earn his PhD at MIT in the Swager lab, where he developed a deep specialization in nanomaterial sensors and field-effect transistors — and more specifically, in how to conceive of novel sensing systems from first principles. That methodology drove the design of Confidynt™: starting from what the sensor needed to do, and working backward to the technology stack capable of doing it.

Prior to Kinovi, Joseph founded Numo Health, where he advanced a novel approach to early disease detection through primary translational research conducted at MGH Cancer Center.

Joseph holds 14 issued patents and 10 pending across US and international jurisdictions. Beyond Kinovi, he works with founders and organizations pursuing consequential problems at the edges of what medicine currently addresses.

Kinovi is an incubator company at the Roux Institute at Northeastern University in Portland, ME, and maintains offices in Boston, MA

Discover with us.

We're building something consequential. If you are too, let's talk.